From: Targeting phosphoglycerate dehydrogenase in multiple myeloma
NCT-503 | ||||||
---|---|---|---|---|---|---|
Cells | Proteosome inhibitor | IC50 of PI | Fold change in IC50 | P value | ||
- NCT | + NCT | |||||
INA6-res | CTR | Carf | 3.6 | 3.2 | 0.89 | 0.1404 |
BTZ | 22.7 | 15.0 | 0.66 | < 0.0001 | ||
CR | Carf | 12.0 | 7.0 | 0.58 | < 0.0001 | |
BTZ | 46.6 | 25.8 | 0.55 | < 0.0001 | ||
BR | Carf | 3.2 | 2.9 | 0.91 | 0.268 | |
BTZ | 59.0 | 34.3 | 0.58 | < 0.0001 | ||
AMO1-res | CTR | Carf | 2.4 | 2.2 | 0.92 | 0.1998 |
BTZ | 24.4 | 7.2 | 0.30 | < 0.0001 | ||
CR | Carf | 711.0 | 645.0 | 0.91 | 0.1521 | |
BTZ | 199.0 | 113.0 | 0.57 | < 0.0001 | ||
BR | Carf | 25.0 | 27.0 | 1.08 | 0.4697 | |
BTZ | 1111.0 | 581.0 | 0.52 | < 0.0001 |